Assay Detail
Functional
CHEMBL802897
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Inhibition of forskolin-stimulated glycogenolysis in SK-HEP-1 cells
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Indole-2-carboxamide inhibitors of human liver glycogen phosphorylase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 5.37 | 5.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL318910 | — | — | 1 | 5.85 |
| CHEMBL319136 | — | — | 1 | 5.82 |
| CHEMBL430503 | — | — | 1 | 5.72 |
| CHEMBL99889 | — | — | 1 | 5.72 |
| CHEMBL327504 | — | — | 1 | 5.64 |
| CHEMBL329493 | — | — | 1 | 5.48 |
| CHEMBL317410 | — | — | 1 | 5.29 |
| CHEMBL99379 | — | — | 1 | 5.28 |
| CHEMBL99597 | — | — | 1 | 5.21 |
| CHEMBL319165 | — | — | 1 | 5.11 |
| CHEMBL98891 | — | — | 1 | 4.92 |
| CHEMBL316598 | — | — | 1 | 4.92 |
| CHEMBL319854 | — | — | 1 | 4.89 |
| CHEMBL319152 | — | — | 1 | - |
| CHEMBL317861 | — | — | 1 | - |
| CHEMBL431463 | — | — | 1 | - |
| CHEMBL100872 | — | — | 1 | - |
| CHEMBL99556 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL318910 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL319136 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL430503 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL99889 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL327504 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL329493 | — | IC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL317410 | — | IC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL99379 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL99597 | — | IC50 | = | 6200.0 | nM | 5.21 |
| CHEMBL319165 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL98891 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL316598 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL319854 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL319152 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL317861 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL431463 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL100872 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL99556 | — | IC50 | > | 30000.0 | nM | - |