Assay Detail
Binding
CHEMBL803151
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Inhibitory activity against human S-adenosyl-L-homocysteine hydrolase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Synthesis of 2-fluoronoraristeromycin and its inhibitory activity against Plasmodium falciparum S-adenosyl-L-homocysteine hydrolase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.08 | 5.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL129014 | NORARISTEROMYCIN | — | 1 | 5.96 |
| CHEMBL129469 | — | — | 1 | 4.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL129014 | NORARISTEROMYCIN | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL129469 | — | IC50 | = | 63000.0 | nM | 4.20 |