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Assay Detail

CHEMBL803155

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards purified recombinant human placental S-adenosyl-L-homocysteine hydrolase
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Adenosylhomocysteinase (CHEMBL2664)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Aristeromycin-5'-carboxaldehyde: a potent inhibitor of S-adenosyl-L-homocysteine hydrolase.
Liu S, Yuan CS, Borchardt RT.
J Med Chem (1996) 39 : 2347 -2353
PubMed 8691429 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 4 6.67 7.41

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL77518 1 7.41
CHEMBL308037 1 7.37
CHEMBL77965 1 6.56
CHEMBL76858 1 5.35

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL77518 Ki = 39.0 nM 7.41
CHEMBL308037 Ki = 43.0 nM 7.37
CHEMBL77965 Ki = 273.0 nM 6.56
CHEMBL76858 Ki = 4500.0 nM 5.35