Assay Detail
Functional
CHEMBL804104
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Ability to reverse NPY-induced intracellular [Ca2+] mobilization in SK-N-MC cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SK-N-MC |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Potent and selective 1,2,3-trisubstituted indole NPY Y-1 antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.49 | 8.49 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL329536 | — | — | 1 | 8.49 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL329536 | — | Ki | = | 3.2 | nM | 8.49 |