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Assay Detail

CHEMBL804128

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibitory activity against bovine liver S-adenosyl-L-homocysteine hydrolase (AdoHcy) rate of inactivation by NpcA
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Bos taurus
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Adenosylhomocysteinase (CHEMBL2664)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

4'-modified analogues of aristeromycin and neplanocin A: synthesis and inhibitory activity toward S-adenosyl-L-homocysteine hydrolase.
Wolfe MS, Lee Y, Bartlett WJ, Borcherding DR, Borchardt RT.
J Med Chem (1992) 35 : 1782 -1791
PubMed 1588558 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.42 8.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL8771 NEOPLANOCIN A 1 8.42

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL8771 NEOPLANOCIN A Ki = 3.8 nM 8.42