Assay Detail
Functional
CHEMBL804749
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Inhibition of Rb negative Skut 1A cell proliferation
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SKUT-1A |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Identification of selective inhibitors of cyclin dependent kinase 4.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.89 | 5.25 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL70713 | — | — | 1 | 5.25 |
| CHEMBL71233 | — | — | 1 | 4.97 |
| CHEMBL71161 | — | — | 1 | 4.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL70713 | — | IC50 | = | 5600.0 | nM | 5.25 |
| CHEMBL71233 | — | IC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL71161 | — | IC50 | = | 36000.0 | nM | 4.44 |