Assay Detail
Binding
CHEMBL804971
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of rhizopuspepsin
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rhizopus microsporus var. chinensis |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Rhizopuspepsin (CHEMBL4253) ↗| Type | SINGLE PROTEIN |
| Organism | Rhizopus microsporus var. chinensis |
Publication
Renin inhibitors. Syntheses of subnanomolar, competitive, transition-state analogue inhibitors containing a novel analogue of statine.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.67 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL269752 | — | — | 1 | 6.70 |
| CHEMBL2028991 | — | — | 1 | 6.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL269752 | — | Ki | = | 200.0 | nM | 6.70 |
| CHEMBL2028991 | — | Ki | = | 230.0 | nM | 6.64 |