Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL805046

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards Somatostatin receptor type 1 (hsst1)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Somatostatin receptor type 1 (CHEMBL1917)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

2002 Alfred Burger Award Address in Medicinal Chemistry. Natural products and design: interrelated approaches in drug discovery.
Patchett AA.
J Med Chem (2002) 45 : 5609 -5616
PubMed 12477342 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 7.52 9.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1823872 SOMATOSTATIN 3.0 1 9.42
CHEMBL99895 1 5.62

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1823872 SOMATOSTATIN Ki = 0.38 nM 9.42
CHEMBL99895 Ki = 2392.0 nM 5.62