Assay Detail
Binding
CHEMBL806598
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Binding affinity for human receptor subtype hSSTR5.
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Modulation of receptor and receptor subtype affinities using diastereomeric and enantiomeric monosaccharide scaffolds as a means to structural and biological diversity. A new route to ether synthesis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 7 | 5.49 | 5.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL282129 | — | — | 1 | 5.89 |
| CHEMBL29102 | — | — | 1 | 5.52 |
| CHEMBL282803 | — | — | 1 | 5.47 |
| CHEMBL282618 | — | — | 1 | 5.43 |
| CHEMBL29311 | — | — | 1 | 5.41 |
| CHEMBL28824 | — | — | 1 | 5.40 |
| CHEMBL281200 | — | — | 1 | 5.29 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL282129 | — | Ki | = | 1300.0 | nM | 5.89 |
| CHEMBL29102 | — | Ki | = | 3000.0 | nM | 5.52 |
| CHEMBL282803 | — | Ki | = | 3400.0 | nM | 5.47 |
| CHEMBL282618 | — | Ki | = | 3700.0 | nM | 5.43 |
| CHEMBL29311 | — | Ki | = | 3900.0 | nM | 5.41 |
| CHEMBL28824 | — | Ki | = | 4000.0 | nM | 5.40 |
| CHEMBL281200 | — | Ki | = | 5100.0 | nM | 5.29 |