Assay Detail
Binding
CHEMBL807058
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The compound was tested for binding affinity against human Somatostatin receptor type 4
40
Total Activities
40
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Highly potent cyclic disulfide antagonists of somatostatin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 40 | 6.09 | 6.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2372960 | — | — | 1 | 6.84 |
| CHEMBL413171 | — | — | 1 | 6.75 |
| CHEMBL439136 | — | — | 1 | 6.52 |
| CHEMBL264028 | — | — | 1 | 6.36 |
| CHEMBL406738 | — | — | 1 | 6.17 |
| CHEMBL2372959 | — | — | 1 | 6.17 |
| CHEMBL410181 | — | — | 1 | 6.14 |
| CHEMBL407496 | — | — | 1 | 6.07 |
| CHEMBL2372964 | — | — | 1 | 6.05 |
| CHEMBL2372961 | — | — | 1 | 6.05 |
| CHEMBL275806 | — | — | 1 | 5.98 |
| CHEMBL408987 | — | — | 1 | 5.80 |
| CHEMBL437220 | — | — | 1 | 5.80 |
| CHEMBL2372957 | — | — | 1 | 5.79 |
| CHEMBL2372956 | — | — | 1 | 5.54 |
| CHEMBL437448 | — | — | 1 | 5.48 |
| CHEMBL384607 | — | — | 1 | - |
| CHEMBL2372963 | — | — | 1 | - |
| CHEMBL411556 | — | — | 1 | - |
| CHEMBL414116 | — | — | 1 | - |
| CHEMBL412859 | — | — | 1 | - |
| CHEMBL408347 | — | — | 1 | - |
| CHEMBL406152 | — | — | 1 | - |
| CHEMBL414386 | — | — | 1 | - |
| CHEMBL408787 | — | — | 1 | - |
| CHEMBL439350 | — | — | 1 | - |
| CHEMBL2372958 | — | — | 1 | - |
| CHEMBL438281 | — | — | 1 | - |
| CHEMBL2372962 | — | — | 1 | - |
| CHEMBL2311098 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2372960 | — | Ki | = | 145.0 | nM | 6.84 |
| CHEMBL413171 | — | Ki | = | 176.0 | nM | 6.75 |
| CHEMBL439136 | — | Ki | = | 301.0 | nM | 6.52 |
| CHEMBL264028 | — | Ki | = | 436.0 | nM | 6.36 |
| CHEMBL406738 | — | Ki | = | 672.0 | nM | 6.17 |
| CHEMBL2372959 | — | Ki | = | 682.0 | nM | 6.17 |
| CHEMBL410181 | — | Ki | = | 728.0 | nM | 6.14 |
| CHEMBL407496 | — | Ki | = | 847.0 | nM | 6.07 |
| CHEMBL2372964 | — | Ki | = | 888.0 | nM | 6.05 |
| CHEMBL2372961 | — | Ki | = | 895.0 | nM | 6.05 |
| CHEMBL275806 | — | Ki | = | 1040.0 | nM | 5.98 |
| CHEMBL408987 | — | Ki | = | 1570.0 | nM | 5.80 |
| CHEMBL437220 | — | Ki | = | 1590.0 | nM | 5.80 |
| CHEMBL2372957 | — | Ki | = | 1640.0 | nM | 5.79 |
| CHEMBL2372956 | — | Ki | = | 2880.0 | nM | 5.54 |
| CHEMBL437448 | — | Ki | = | 3310.0 | nM | 5.48 |
| CHEMBL385746 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL412561 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL264539 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL414598 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL439005 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL407195 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL406491 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL413709 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL415201 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL385689 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL2311098 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL2372962 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL438281 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL2372958 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL439350 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL408787 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL414386 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL406152 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL408347 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL412859 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL414116 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL411556 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL2372963 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL384607 | — | Ki | > | 1000.0 | nM | - |