Assay Detail
Binding
CHEMBL808445
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Compound was tested for inhibition against tissue factor.
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Pyrazoles, 1,2,4-triazoles, and tetrazoles as surrogates for cis-amide bonds in boronate ester thrombin inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.86 | 6.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2373367 | — | — | 1 | 6.17 |
| CHEMBL2373345 | — | — | 1 | 5.55 |
| CHEMBL2373400 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2373367 | — | Ki | = | 670.0 | nM | 6.17 |
| CHEMBL2373345 | — | Ki | = | 2800.0 | nM | 5.55 |
| CHEMBL2373400 | — | Ki | > | 10000.0 | nM | - |