Assay Detail

CHEMBL810204

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional

Tested for its binding effect on [3H]- DAMGO in bovine striatal membrane at 20 nM

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Bos taurus
Tissue	Striatum
Subcellular	Membrane
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

14 beta-[(p-nitrocinnamoyl)amino]morphinones, 14 beta-[(p-nitrocinnamoyl)amino]-7,8-dihydromorphinones, and their codeinone analogues: synthesis and receptor activity.

Sebastian A, Bidlack JM, Jiang Q, Deecher D, Teitler M, Glick SD, Archer S.
J Med Chem (1993) 36 : 3154 -3160
PubMed 7693944 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
Kd	1	9.09	9.09

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL108406	—	—	1	9.09

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL108406	—	Kd	=	0.82	nM	9.09