Assay Detail
Binding
CHEMBL810718
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Inhibitory activity against Selectin P IgG chimera binding to HL-60 cells, by binding to Selectin P
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | HL-60 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Carbohydrates in an acidic multivalent assembly: nanomolar P-selectin inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.50 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2303775 | — | — | 1 | 8.70 |
| CHEMBL7864 | — | — | 1 | 6.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2303775 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL7864 | — | IC50 | = | 500.0 | nM | 6.30 |