Assay Detail
Binding
CHEMBL810833
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Inhibitory activity against Serum amine oxidase
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 4.63 | 5.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL120717 | — | — | 1 | 5.26 |
| CHEMBL121432 | — | — | 1 | 5.00 |
| CHEMBL331009 | — | — | 1 | 4.24 |
| CHEMBL331650 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL120717 | — | Ki | = | 5500.0 | nM | 5.26 |
| CHEMBL121432 | — | Ki | = | 10000.0 | nM | 5.00 |
| CHEMBL331009 | — | Ki | = | 57000.0 | nM | 4.24 |
| CHEMBL331650 | — | Ki | = | 100000.0 | nM | 4.00 |