Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL811862

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for inhibition of tryptase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Tryptase gamma (CHEMBL4955)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

3-Amidinophenylalanine-based inhibitors of urokinase.
Stürzebecher J, Vieweg H, Steinmetzer T, Schweinitz A, Stubbs MT, Renatus M, Wikström P.
Bioorg Med Chem Lett (1999) 9 : 3147 -3152
PubMed 10560742 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.20 5.20

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL107955 1 5.20

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL107955 Ki = 6300.0 nM 5.20