Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL815305

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Effective concentration (EC50) required to inhibit UT7/TPO Cell Proliferation was determined.
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Hydrazinonaphthalene and azonaphthalene thrombopoietin mimics are nonpeptidyl promoters of megakaryocytopoiesis.
Duffy KJ, Darcy MG, Delorme E, Dillon SB, Eppley DF, Erickson-Miller C, Giampa L, Hopson CB, Huang Y, Keenan RM, Lamb P, Leong L, Liu N, Miller SG, Price AT, Rosen J, Shah R, Shaw TN, Smith H, Stark KC, Tian SS, Tyree C, Wiggall KJ, Zhang L, Luengo JI.
J Med Chem (2001) 44 : 3730 -3745
PubMed 11606138 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 6.59 7.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3144844 1 7.16
CHEMBL3144789 1 6.30
CHEMBL3144852 1 6.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3144844 EC50 = 70.0 nM 7.16
CHEMBL3144789 EC50 = 500.0 nM 6.30
CHEMBL3144852 EC50 = 500.0 nM 6.30