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Assay Detail

CHEMBL815426

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Mn2+ activated state of very late antigen 4 (VLA-4)
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 6 — Multiple protein complex / RNA
Curated By Autocuration

Target

Integrin alpha-4/beta-1 (CHEMBL1907599)
Type PROTEIN COMPLEX
Organism Homo sapiens

Publication

Bioisosteric replacement of anilide with benzoxazole: potent and orally bioavailable antagonists of VLA-4.
Lin LS, Lanza TJ, Castonguay LA, Kamenecka T, McCauley E, Van Riper G, Egger LA, Mumford RA, Tong X, MacCoss M, Schmidt JA, Hagmann WK.
Bioorg Med Chem Lett (2004) 14 : 2331 -2334
PubMed 15081035 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 9.33 10.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL309823 1 10.15
CHEMBL73986 1 9.57
CHEMBL77586 1 9.47
CHEMBL76295 1 9.27
CHEMBL306739 1 9.16
CHEMBL77924 1 9.13
CHEMBL308346 1 9.10
CHEMBL265778 1 8.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL309823 IC50 = 0.07 nM 10.15
CHEMBL73986 IC50 = 0.27 nM 9.57
CHEMBL77586 IC50 = 0.34 nM 9.47
CHEMBL76295 IC50 = 0.54 nM 9.27
CHEMBL306739 IC50 = 0.69 nM 9.16
CHEMBL77924 IC50 = 0.74 nM 9.13
CHEMBL308346 IC50 = 0.79 nM 9.10
CHEMBL265778 IC50 = 1.7 nM 8.77