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Assay Detail

CHEMBL815568

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxic concentration against Vero cells was determined on day 3
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Chlorocebus sabaeus
Cell Type Vero
Confidence 1 — Organism
Curated By Intermediate

Target

Vero (CHEMBL391)
Type CELL-LINE
Organism Chlorocebus sabaeus

Publication

Synthesis and biological properties of 5-o-carboranyl-1-(2-deoxy-2-fluoro-beta-D-arabinofuranosyl)uracil.
Fulcrand-el Kattan G, Goudgaon NM, Ilksoy N, Huang JT, Watanabe KA, Sommadossi JP, Schinazi RF.
J Med Chem (1994) 37 : 2583 -2588
PubMed 8057301 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.56 4.76

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3142561 1 4.76
CHEMBL129 ZIDOVUDINE 4.0 1 4.54
CHEMBL3142559 1 4.39

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3142561 IC50 = 17300.0 nM 4.76
CHEMBL129 ZIDOVUDINE IC50 = 29000.0 nM 4.54
CHEMBL3142559 IC50 = 41100.0 nM 4.39