Assay Detail

CHEMBL818549

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional

Inhibition of [3H]-BTX binding to cardiac voltage-gated sodium channel

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Rattus norvegicus
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Medicinal chemistry of neuronal voltage-gated sodium channel blockers.

Anger T, Madge DJ, Mulla M, Riddall D.
J Med Chem (2001) 44 : 115 -137
PubMed 11170622 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	6.00	6.00

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL29404	ENECADIN	2.0	1	6.00

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL29404	ENECADIN	IC50	=	1000.0	nM	6.00