Assay Detail
Functional
CHEMBL819025
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Tested in vitro for effective concentration required for stimulation of phospholipase C (PLC) against [3H]inositol labeled Turkey Erythrocyte P2Y purinoceptor 1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Meleagris gallopavo |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Acyclic analogues of deoxyadenosine 3',5'-bisphosphates as P2Y(1) receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.17 | 5.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1230817 | — | — | 1 | 5.20 |
| CHEMBL165225 | — | — | 1 | 5.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1230817 | — | EC50 | = | 6290.0 | nM | 5.20 |
| CHEMBL165225 | — | EC50 | = | 7210.0 | nM | 5.14 |