Assay Detail
Binding
CHEMBL820157
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro binding affinity towards alpha-adreno ceptor of rat forebrain using [3H]prazosin
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Synthesis and biological properties of thiophene ring analogues of mianserin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.19 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL13644 | — | — | 1 | 6.52 |
| CHEMBL13645 | — | — | 1 | 5.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL13644 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL13645 | — | IC50 | = | 1400.0 | nM | 5.85 |