Assay Detail
Binding
CHEMBL821730
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Inhibitory activity against calpain.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Protease inhibitors: current status and future prospects.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.78 | 7.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL115073 | — | — | 1 | 7.55 |
| CHEMBL92708 | CALPEPTIN | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL115073 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL92708 | CALPEPTIN | IC50 | = | 1000.0 | nM | 6.00 |