Assay Detail
Binding
CHEMBL823703
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Compound was tested for inhibition of specific [3H]cantharidin binding to CBP: Range= 10-50
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of protein phosphatase 2A by cantharidin analogues
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.30 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL8182 | — | — | 1 | 7.30 |
| CHEMBL273884 | — | — | 1 | 7.30 |
| CHEMBL428650 | ENDOTHALL | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL8182 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL273884 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL428650 | ENDOTHALL | IC50 | = | 50.0 | nM | 7.30 |