Assay Detail
Binding
CHEMBL826979
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Inhibitory concentration against Platelet-derived growth factor receptor
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Substituted aminobenzimidazole pyrimidines as cyclin-dependent kinase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 6.93 | 7.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL372464 | — | — | 1 | 7.48 |
| CHEMBL195641 | — | — | 1 | 6.96 |
| CHEMBL364935 | — | — | 1 | 6.72 |
| CHEMBL194721 | — | — | 1 | 6.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL372464 | — | IC50 | = | 33.0 | nM | 7.48 |
| CHEMBL195641 | — | IC50 | = | 110.0 | nM | 6.96 |
| CHEMBL364935 | — | IC50 | = | 190.0 | nM | 6.72 |
| CHEMBL194721 | — | IC50 | = | 290.0 | nM | 6.54 |