Assay Detail
Binding
CHEMBL826997
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro dissociation constant for heat shock 90 kDa protein alpha
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Crystal structures of human HSP90alpha-complexed with dihydroxyphenylpyrazoles.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.36 | 6.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL360563 | — | — | 1 | 6.55 |
| CHEMBL178130 | — | — | 1 | 6.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL360563 | — | Kd | = | 280.0 | nM | 6.55 |
| CHEMBL178130 | — | Kd | = | 680.0 | nM | 6.17 |