Assay Detail
Functional
CHEMBL827419
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Mitogenic stimulation or antagonism of 30 nM quinpirole-stimulated mitogenesis in CHO cells expressing human dopamine D2 receptor
17
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Dopamine D3 receptor partial agonists and antagonists as potential drug abuse therapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 7.24 | 8.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL71865 | — | — | 1 | 8.13 |
| CHEMBL195057 | — | — | 1 | 8.08 |
| CHEMBL194493 | — | — | 1 | 7.86 |
| CHEMBL301242 | — | — | 2 | 7.84 |
| CHEMBL71327 | — | — | 1 | 7.79 |
| CHEMBL302374 | — | — | 1 | 7.26 |
| CHEMBL370713 | — | — | 1 | 7.21 |
| CHEMBL262724 | — | — | 1 | 7.12 |
| CHEMBL180010 | — | — | 1 | 7.09 |
| CHEMBL69451 | — | — | 1 | 7.04 |
| CHEMBL59725 | — | — | 1 | 7.02 |
| CHEMBL366904 | — | — | 1 | 6.96 |
| CHEMBL139926 | — | — | 1 | 6.93 |
| CHEMBL180060 | — | — | 1 | 6.79 |
| CHEMBL175734 | — | — | 1 | 6.59 |
| CHEMBL300780 | — | — | 1 | 5.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL71865 | — | IC50 | = | 7.49 | nM | 8.13 |
| CHEMBL195057 | — | IC50 | = | 8.29 | nM | 8.08 |
| CHEMBL194493 | — | IC50 | = | 13.8 | nM | 7.86 |
| CHEMBL301242 | — | IC50 | = | 14.6 | nM | 7.84 |
| CHEMBL71327 | — | IC50 | = | 16.1 | nM | 7.79 |
| CHEMBL301242 | — | IC50 | = | 35.6 | nM | 7.45 |
| CHEMBL302374 | — | IC50 | = | 55.4 | nM | 7.26 |
| CHEMBL370713 | — | IC50 | = | 61.8 | nM | 7.21 |
| CHEMBL262724 | — | IC50 | = | 76.7 | nM | 7.12 |
| CHEMBL180010 | — | IC50 | = | 80.9 | nM | 7.09 |
| CHEMBL69451 | — | IC50 | = | 92.0 | nM | 7.04 |
| CHEMBL59725 | — | IC50 | = | 94.7 | nM | 7.02 |
| CHEMBL366904 | — | IC50 | = | 111.0 | nM | 6.96 |
| CHEMBL139926 | — | IC50 | = | 118.0 | nM | 6.93 |
| CHEMBL180060 | — | IC50 | = | 162.0 | nM | 6.79 |
| CHEMBL175734 | — | IC50 | = | 254.0 | nM | 6.59 |
| CHEMBL300780 | — | IC50 | = | 1280.0 | nM | 5.89 |