Assay Detail
Binding
CHEMBL828012
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Inhibition of [125I]IABN binding to human Dopamine D3 receptor expressed in HEK 293 cells
18
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Dopamine D3 receptor partial agonists and antagonists as potential drug abuse therapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 18 | 8.74 | 9.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL71865 | — | — | 1 | 9.40 |
| CHEMBL195057 | — | — | 1 | 9.40 |
| CHEMBL69451 | — | — | 1 | 9.30 |
| CHEMBL180010 | — | — | 1 | 9.15 |
| CHEMBL194493 | — | — | 1 | 9.15 |
| CHEMBL59725 | — | — | 1 | 9.10 |
| CHEMBL71327 | — | — | 1 | 9.10 |
| CHEMBL139926 | — | — | 1 | 9.10 |
| CHEMBL175734 | — | — | 2 | 8.96 |
| CHEMBL370713 | — | — | 1 | 8.92 |
| CHEMBL262724 | — | — | 1 | 8.85 |
| CHEMBL302374 | — | — | 1 | 8.80 |
| CHEMBL300780 | — | — | 1 | 8.70 |
| CHEMBL366904 | — | — | 1 | 8.68 |
| CHEMBL180060 | — | — | 1 | 8.47 |
| CHEMBL301242 | — | — | 1 | 8.40 |
| CHEMBL69571 | — | — | 1 | 8.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL195057 | — | Ki | = | 0.4 | nM | 9.40 |
| CHEMBL71865 | — | Ki | = | 0.4 | nM | 9.40 |
| CHEMBL69451 | — | Ki | = | 0.5 | nM | 9.30 |
| CHEMBL180010 | — | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL194493 | — | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL59725 | — | Ki | = | 0.8 | nM | 9.10 |
| CHEMBL139926 | — | Ki | = | 0.8 | nM | 9.10 |
| CHEMBL71327 | — | Ki | = | 0.8 | nM | 9.10 |
| CHEMBL175734 | — | Ki | = | 1.1 | nM | 8.96 |
| CHEMBL370713 | — | Ki | = | 1.2 | nM | 8.92 |
| CHEMBL262724 | — | Ki | = | 1.4 | nM | 8.85 |
| CHEMBL302374 | — | Ki | = | 1.6 | nM | 8.80 |
| CHEMBL300780 | — | Ki | = | 2.0 | nM | 8.70 |
| CHEMBL366904 | — | Ki | = | 2.1 | nM | 8.68 |
| CHEMBL180060 | — | Ki | = | 3.4 | nM | 8.47 |
| CHEMBL301242 | — | Ki | = | 4.0 | nM | 8.40 |
| CHEMBL69571 | — | Ki | = | 8.2 | nM | 8.09 |
| CHEMBL175734 | — | Ki | = | 1770.0 | nM | 5.75 |