Assay Detail
Binding
CHEMBL828050
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Inhibitory concentration for human liver monoamine oxidase B
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Fluorinated phenylcyclopropylamines. 2. Effects of aromatic ring substitution and of absolute configuration on inhibition of microbial tyramine oxidase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.02 | 5.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2093956 | — | — | 1 | 5.17 |
| CHEMBL903 | HYDRAZINECARBOXAMIDE | — | 1 | 5.17 |
| CHEMBL542118 | — | — | 1 | 4.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2093956 | — | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL903 | HYDRAZINECARBOXAMIDE | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL542118 | — | IC50 | = | 19000.0 | nM | 4.72 |