Assay Detail
Binding
CHEMBL828061
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Inhibition of 5-hydroxytryptamine 1D receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Indolebutylamines as selective 5-HT(1A) agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.28 | 6.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL363537 | — | — | 1 | 6.40 |
| CHEMBL360419 | — | — | 1 | 6.16 |
| CHEMBL187196 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL363537 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL360419 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL187196 | — | IC50 | > | 1000.0 | nM | - |