Assay Detail
Binding
CHEMBL828064
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of 5-hydroxytryptamine 2A receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of CC chemokine receptor-3 (CCR3) antagonists with picomolar potency.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.80 | 6.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL250689 | — | — | 1 | 6.04 |
| CHEMBL195433 | — | — | 1 | 5.85 |
| CHEMBL363840 | — | — | 1 | 5.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL250689 | — | IC50 | = | 920.0 | nM | 6.04 |
| CHEMBL195433 | — | IC50 | = | 1415.0 | nM | 5.85 |
| CHEMBL363840 | — | IC50 | = | 3120.0 | nM | 5.51 |