Assay Detail
Binding
CHEMBL828169
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition concentration against tyramine oxidase of Arthrobacter spp.; Partially irreversible inhibition
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Fluorinated phenylcyclopropylamines. 2. Effects of aromatic ring substitution and of absolute configuration on inhibition of microbial tyramine oxidase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.09 | 4.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2094041 | — | — | 1 | 4.12 |
| CHEMBL541373 | — | — | 1 | 4.05 |
| CHEMBL2093957 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2094041 | — | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL541373 | — | IC50 | = | 89000.0 | nM | 4.05 |
| CHEMBL2093957 | — | IC50 | = | 190000.0 | nM | - |