Assay Detail
Binding
CHEMBL828250
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Binding affinity against rabbit muscle triose-phosphate isomerase
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Tissue | Muscle tissue |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
New inhibitors of rabbit muscle triose-phosphate isomerase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.44 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL371668 | PHOSPHOGLYCOLOHYDROXAMATE | — | 1 | 5.52 |
| CHEMBL195976 | — | — | 1 | 5.35 |
| CHEMBL195520 | PHOSPHORIC ACID MONOHYDRAZINOCARBONYLMETHYL ESTER | — | 1 | - |
| CHEMBL196442 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL371668 | PHOSPHOGLYCOLOHYDROXAMATE | Ki | = | 3000.0 | nM | 5.52 |
| CHEMBL195976 | — | Ki | = | 4500.0 | nM | 5.35 |
| CHEMBL195520 | PHOSPHORIC ACID MONOHYDRAZINOCARBONYLMETHYL ESTER | Ki | = | 111000.0 | nM | - |
| CHEMBL196442 | — | Ki | = | 159000.0 | nM | - |