Assay Detail
Binding
CHEMBL828788
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition constant against luciferase with respect to luciferyl-adenylate
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Luciola lateralis |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis of an N-acyl sulfamate analog of luciferyl-AMP: a stable and potent inhibitor of firefly luciferase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.47 | 6.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1235965 | — | — | 1 | 6.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1235965 | — | Ki | = | 340.0 | nM | 6.47 |