Assay Detail
Binding
CHEMBL828804
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]CP-55940 binding to cannabinoid receptor 1 of rat brain
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Adamantyl cannabinoids: a novel class of cannabinergic ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 6 | 7.48 | 8.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL434351 | — | — | 1 | 8.17 |
| CHEMBL480107 | — | — | 1 | 7.53 |
| CHEMBL371167 | — | — | 1 | 7.46 |
| CHEMBL267227 | DELTA-8-TETRAHYDROCANNABINOL | 2.0 | 1 | 7.32 |
| CHEMBL191324 | — | — | 1 | 7.31 |
| CHEMBL372866 | — | — | 1 | 7.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL434351 | — | Ki | = | 6.8 | nM | 8.17 |
| CHEMBL480107 | — | Ki | = | 29.3 | nM | 7.53 |
| CHEMBL371167 | — | Ki | = | 34.9 | nM | 7.46 |
| CHEMBL267227 | DELTA-8-TETRAHYDROCANNABINOL | Ki | = | 47.6 | nM | 7.32 |
| CHEMBL191324 | — | Ki | = | 48.6 | nM | 7.31 |
| CHEMBL372866 | — | Ki | = | 79.7 | nM | 7.10 |