Assay Detail
Binding
CHEMBL828827
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]PGE-2 binding to Prostanoid EP2 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Prostaglandin E2 receptor EP2 subtype (CHEMBL1881) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Metabolism investigation leading to novel drug design: orally active prostacyclin mimetics. Part 4.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.85 | 5.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2373410 | — | — | 1 | 5.85 |
| CHEMBL132589 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2373410 | — | Ki | = | 1400.0 | nM | 5.85 |
| CHEMBL132589 | — | Ki | > | 1000.0 | nM | - |