Assay Detail
Binding
CHEMBL828890
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Inhibition of [3H]YM-09151-2 binding to human Dopamine D2L receptor expressed in CHO cells
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Dopamine D3 receptor partial agonists and antagonists as potential drug abuse therapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 18 | 7.14 | 7.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL71865 | — | — | 1 | 7.82 |
| CHEMBL301242 | — | — | 1 | 7.71 |
| CHEMBL71327 | — | — | 1 | 7.63 |
| CHEMBL194493 | — | — | 1 | 7.51 |
| CHEMBL59725 | — | — | 1 | 7.37 |
| CHEMBL302374 | — | — | 1 | 7.29 |
| CHEMBL262724 | — | — | 1 | 7.23 |
| CHEMBL69451 | — | — | 1 | 7.21 |
| CHEMBL195057 | — | — | 1 | 7.18 |
| CHEMBL370713 | — | — | 1 | 7.01 |
| CHEMBL180010 | — | — | 1 | 6.97 |
| CHEMBL139926 | — | — | 1 | 6.92 |
| CHEMBL366904 | — | — | 1 | 6.88 |
| CHEMBL180060 | — | — | 1 | 6.72 |
| CHEMBL175734 | — | — | 1 | 6.61 |
| CHEMBL300780 | — | — | 1 | 6.16 |
| CHEMBL69571 | — | — | 1 | - |
| CHEMBL304605 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL71865 | — | Ki | = | 15.2 | nM | 7.82 |
| CHEMBL301242 | — | Ki | = | 19.4 | nM | 7.71 |
| CHEMBL71327 | — | Ki | = | 23.4 | nM | 7.63 |
| CHEMBL194493 | — | Ki | = | 31.0 | nM | 7.51 |
| CHEMBL59725 | — | Ki | = | 42.5 | nM | 7.37 |
| CHEMBL302374 | — | Ki | = | 51.4 | nM | 7.29 |
| CHEMBL262724 | — | Ki | = | 58.3 | nM | 7.23 |
| CHEMBL69451 | — | Ki | = | 61.2 | nM | 7.21 |
| CHEMBL195057 | — | Ki | = | 65.8 | nM | 7.18 |
| CHEMBL370713 | — | Ki | = | 96.5 | nM | 7.01 |
| CHEMBL180010 | — | Ki | = | 106.0 | nM | 6.97 |
| CHEMBL139926 | — | Ki | = | 119.0 | nM | 6.92 |
| CHEMBL366904 | — | Ki | = | 131.0 | nM | 6.88 |
| CHEMBL180060 | — | Ki | = | 192.0 | nM | 6.72 |
| CHEMBL175734 | — | Ki | = | 245.0 | nM | 6.61 |
| CHEMBL300780 | — | Ki | = | 698.0 | nM | 6.16 |
| CHEMBL69571 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL304605 | — | Ki | > | 10000.0 | nM | - |