Assay Detail
Binding
CHEMBL829240
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Inhibition of Cyclin-dependent kinase 2
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Conformation mining: an algorithm for finding biologically relevant conformations.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 7.00 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1276446 | — | — | 1 | 8.00 |
| CHEMBL102926 | — | — | 1 | 8.00 |
| CHEMBL101311 | — | — | 1 | 6.00 |
| CHEMBL191845 | — | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1276446 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL102926 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL101311 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL191845 | — | IC50 | = | 1000.0 | nM | 6.00 |