Assay Detail
Binding
CHEMBL829533
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of trypsin like activity of the proteasome in colon carcinoma cell lines COO115
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 2 — Organism |
| Curated By | Expert |
Publication
Peptidyl vinyl ester derivatives: new class of selective inhibitors of proteasome trypsin-like activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.39 | 7.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL189919 | — | — | 1 | 7.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL189919 | — | IC50 | = | 41.0 | nM | 7.39 |