Assay Detail
Binding
CHEMBL830347
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Binding affinity against human sst5 receptor at a dose of 10 uM
3
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 9.52 | 9.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1823872 | SOMATOSTATIN | 3.0 | 3 | 9.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1823872 | SOMATOSTATIN | Ki | = | 0.15 | nM | 9.82 |
| CHEMBL1823872 | SOMATOSTATIN | Ki | = | 0.26 | nM | 9.59 |
| CHEMBL1823872 | SOMATOSTATIN | Ki | = | 0.71 | nM | 9.15 |