Assay Detail
Binding
CHEMBL832754
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory effect on 20S proteasome chymotrypsin-like activity
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 2 — Organism |
| Curated By | Expert |
Publication
Retro hydrazino-azapeptoids as peptidomimetics of proteasome inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.82 | 4.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL304784 | — | — | 1 | 4.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL304784 | — | IC50 | = | 15000.0 | nM | 4.82 |