Assay Detail
Functional
CHEMBL832967
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory concentration was measured against B16 (melanoma) cell from mouse at 24 hours
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | B16 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
N1-substituent effects in the selective delivery of polyamine conjugates into cells containing active polyamine transporters.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.22 | 5.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL541629 | — | — | 1 | 5.72 |
| CHEMBL555288 | — | — | 1 | 4.71 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL541629 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL555288 | — | IC50 | = | 19300.0 | nM | 4.71 |