Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL833115

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Effective concentration to induce a quorum signal in Vibrio harveyi(by binding Lux P protein)
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vibrio harveyi
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Quorum sensing in Vibrio harveyi: probing the specificity of the LuxP binding site.
Lowery CA, McKenzie KM, Qi L, Meijler MM, Janda KD.
Bioorg Med Chem Lett (2005) 15 : 2395 -2398
PubMed 15837332 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 8 5.11 7.36

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL193493 1 7.36
CHEMBL193495 1 4.57
CHEMBL193817 1 4.41
CHEMBL194166 1 4.08
CHEMBL193424 1 -
CHEMBL195989 1 -
CHEMBL195094 1 -
CHEMBL196 ASCORBIC ACID 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL193493 EC50 = 44.0 nM 7.36
CHEMBL193495 EC50 = 27000.0 nM 4.57
CHEMBL193817 EC50 = 39000.0 nM 4.41
CHEMBL194166 EC50 = 84000.0 nM 4.08
CHEMBL193424 EC50 = 429000.0 nM -
CHEMBL195989 EC50 = 108000.0 nM -
CHEMBL195094 EC50 = 560000.0 nM -
CHEMBL196 ASCORBIC ACID EC50 = 737000.0 nM -