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Assay Detail

CHEMBL833395

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Compound was tested for the inhibition of HCV NS5B-mediated RNA synthesis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Intermediate

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Structure-activity relationship of heterobase-modified 2'-C-methyl ribonucleosides as inhibitors of hepatitis C virus RNA replication.
Eldrup AB, Prhavc M, Brooks J, Bhat B, Prakash TP, Song Q, Bera S, Bhat N, Dande P, Cook PD, Bennett CF, Carroll SS, Ball RG, Bosserman M, Burlein C, Colwell LF, Fay JF, Flores OA, Getty K, LaFemina RL, Leone J, MacCoss M, McMasters DR, Tomassini JE, Von Langen D, Wolanski B, Olsen DB.
J Med Chem (2004) 47 : 5284 -5297
PubMed 15456273 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.31 6.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL418899 2'-B-METHYL-GUANOSINE 1 6.89
CHEMBL73809 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL418899 2'-B-METHYL-GUANOSINE IC50 = 130.0 nM 6.89
CHEMBL73809 IC50 = 1900.0 nM 5.72