Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL833551

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibitory concentration against alpha-galactosidase of coffee bean
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Coffea arabica
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Biological properties of D- and L-1-deoxyazasugars.
Kato A, Kato N, Kano E, Adachi I, Ikeda K, Yu L, Okamoto T, Banba Y, Ouchi H, Takahata H, Asano N.
J Med Chem (2005) 48 : 2036 -2044
PubMed 15771446 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.86 8.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL110458 MIGALASTAT 4.0 1 8.52
CHEMBL176021 1 4.89
CHEMBL368121 1 4.17
CHEMBL307429 DUVOGLUSTAT 2.0 1 -
CHEMBL176206 1 -
CHEMBL179130 1 -
CHEMBL369046 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL110458 MIGALASTAT IC50 = 3.0 nM 8.52
CHEMBL176021 IC50 = 13000.0 nM 4.89
CHEMBL368121 IC50 = 67000.0 nM 4.17
CHEMBL307429 DUVOGLUSTAT IC50 = 880000.0 nM -
CHEMBL176206 IC50 = 260000.0 nM -
CHEMBL179130 IC50 = 290000.0 nM -
CHEMBL369046 IC50 = 160000.0 nM -