Assay Detail
Functional
CHEMBL836174
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Equilibrium constant of compound for binding to the active sites in human PC-3 cell membranes
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PC-3 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Potent bombesin-like peptides for GRP-receptor targeting of tumors with 99mTc: a preclinical study.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 10.00 | 10.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL414307 | — | — | 1 | 10.15 |
| CHEMBL266079 | — | — | 1 | 9.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL414307 | — | Kd | = | 0.07 | nM | 10.15 |
| CHEMBL266079 | — | Kd | = | 0.14 | nM | 9.85 |