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Assay Detail

CHEMBL840078

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity for the recombinant XIAP BIR3 protein in displacing a fluorescently labeled Smac peptide
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

E3 ubiquitin-protein ligase XIAP (CHEMBL4198)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structure-based design, synthesis, and evaluation of conformationally constrained mimetics of the second mitochondria-derived activator of caspase that target the X-linked inhibitor of apoptosis protein/caspase-9 interaction site.
Sun H, Nikolovska-Coleska Z, Yang CY, Xu L, Tomita Y, Krajewski K, Roller PP, Wang S.
J Med Chem (2004) 47 : 4147 -4150
PubMed 15293984 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 11 5.64 6.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL534477 1 6.54
CHEMBL535596 1 6.46
CHEMBL365059 1 6.24
CHEMBL534922 1 5.85
CHEMBL556818 1 5.63
CHEMBL536268 1 5.35
CHEMBL536038 1 4.65
CHEMBL557362 1 4.37
CHEMBL558170 1 -
CHEMBL537185 1 -
CHEMBL538075 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL534477 Ki = 290.0 nM 6.54
CHEMBL535596 Ki = 350.0 nM 6.46
CHEMBL365059 Ki = 580.0 nM 6.24
CHEMBL534922 Ki = 1410.0 nM 5.85
CHEMBL556818 Ki = 2330.0 nM 5.63
CHEMBL536268 Ki = 4470.0 nM 5.35
CHEMBL536038 Ki = 22400.0 nM 4.65
CHEMBL557362 Ki = 43110.0 nM 4.37
CHEMBL558170 Ki > 100000.0 nM -
CHEMBL537185 Ki > 100000.0 nM -
CHEMBL538075 Ki > 100000.0 nM -