Assay Detail
Binding
CHEMBL841023
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranes
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | PC-12 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.72 | 7.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL275970 | TRACIZOLINE | — | 1 | 7.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL275970 | TRACIZOLINE | Ki | = | 19.05 | nM | 7.72 |