Assay Detail
Binding
CHEMBL841025
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Binding affinity at imidazoline receptor I-1 of rat.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Binding of beta-carbolines at imidazoline I2 receptors: a structure-affinity investigation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.43 | 5.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL6857 | — | — | 1 | 5.43 |
| CHEMBL6310 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL6857 | — | Ki | = | 3740.0 | nM | 5.43 |
| CHEMBL6310 | — | Ki | > | 100000.0 | nM | - |