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Assay Detail

CHEMBL842650

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards r5HT2 receptor.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Serotonin 2 (5-HT2) receptor (CHEMBL2093870)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Current and novel approaches to the drug treatment of schizophrenia.
Rowley M, Bristow LJ, Hutson PH.
J Med Chem (2001) 44 : 477 -501
PubMed 11170639 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.59 9.59

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL83894 FANANSERIN 2.0 1 9.59

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL83894 FANANSERIN Ki = 0.26 nM 9.59