Assay Detail
Functional
CHEMBL843249
Review assay metadata, readout intent, target linkage, and publication context from the same page.
The compound (synthetic) was tested for the ability to inhibit inducible cell adhesion molecule expression (E-selectin) in primary human endothelial cell line (HUVEC)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HUVEC |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Synthesis and evaluation of aza HUN-7293.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.00 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2448563 | — | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2448563 | — | IC50 | = | 1000.0 | nM | 6.00 |